51
2
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T22538 |
A-7 hydrochloride
|
CaMK | Neuroscience |
A-7 hydrochloride 是一种钙调蛋白拮抗剂,会引起 MDA-MB-231细胞中 CD44+CD24-亚群的改变。 | |||
T11638 |
Ilorasertib hydrochloride
ABT-348 hydrochloride |
Aurora Kinase | Cell Cycle/Checkpoint; Chromatin/Epigenetic |
Ilorasertib hydrochloride (ABT-348 hydrochloride) is an ATP-competitive multitargeted kinase inhibitor, which inhibits Aurora C, Aurora B, and Aurora A (IC50s: 1 nM, 7 nM, 120 nM). It also suppresses RET tyrosine kinase, PDGFRβ, and Flt1 (IC50s: 7 nM, 3 nM, and 32 nM). | |||
T4690 |
Betrixaban hydrochloride(330942-05-7(free base))
PRT054021 hydrochloride,盐酸贝曲西班 |
Factor Xa | Metabolism |
Betrixaban hydrochloride(330942-05-7(free base)) (PRT054021 hydrochloride) 是一种有效的、选择性的、口服有效的 Xa 因子 (fXa) 抑制剂 (IC50: 1.5 nM)。 | |||
T20792 |
W-7 hydrochloride
N-(6-氨基己基)-5-氯-1-萘磺胺盐酸盐,W 7 HCl,W7 HCl,W-7 HCl |
CaMK; Apoptosis; Myosin; PDE | Apoptosis; Cytoskeletal Signaling; Metabolism; Neuroscience |
W-7 hydrochloride (W-7 HCl) 是一种选择性的钙调蛋白拮抗剂。它抑制Ca2+-钙调蛋白依赖性磷酸二酯酶和肌球蛋白轻链激酶,IC50值分别为 28 μM 和 51 μM。它可诱导细胞凋亡,具有抗癌活性。 | |||
T28531 |
Facinicline hydrochloride
RG3487 |
5-HT Receptor; AChR | GPCR/G Protein; Neuroscience |
Facinicline hydrochloride (RG3487) 是一种口服有效的烟碱α7 receptor 部分激动剂,对人 nAChR 的 Ki 值为 6 nM。它可改善啮齿类动物的认知和感觉运动门控。它与5-HT3受体结合的 Ki 为 1.2 nM。 | |||
T3050 |
ML-7 hydrochloride
ML-7 HCl,ML-7盐酸盐 |
Serine/threonin kinase; Myosin; YAP; PKA; PKC | Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; Metabolism; Stem Cells; Tyrosine Kinase/Adaptors |
ML-7 hydrochloride (ML-7 HCl) 是一种可渗透细胞的、可逆的、有效的、ATP 竞争性的肌球蛋白轻链激酶(MLCK) 特异性抑制剂,IC50为300 nM。它还抑制平滑肌肌球蛋白轻链激酶、PKA 和 PKC。 | |||
T10883L |
CRA-026440 hydrochloride
CRA-026440 hydrochloride(847460-34-8 Free base) |
HDAC | Chromatin/Epigenetic; DNA Damage/DNA Repair |
CRA-026440 hydrochloride 是有效的、广谱的 HDAC 抑制剂。CRA-026440 hydrochloride 作用于 HDAC1,HDAC2,HDAC3,HDAC6,HDAC8 和 HDAC10, Ki 值分别为 4 nM,14 nM,11 nM,15 nM,7 nM 和 20 nM。CRA-026440 hydrochloride 具有抗血管生成和抗肿瘤活性。 | |||
T11719 |
JMV 2959 hydrochloride (925238-89-7 free base)
JMV 2959 hydrochloride |
GHSR | GPCR/G Protein |
JMV 2959 hydrochloride (925238-89-7 free base) 是一种生长激素促分泌素受体 1a 型 (GHS-R1a) 拮抗剂,在 LLC-PK1 细胞中的 IC50 为 32±3 nM。 | |||
T5164 |
Cabozantinib hydrochloride
XL184,Cabozantinib hydrochloride (849217-68-1(free base)),BMS-907351,盐酸卡博替尼 |
VEGFR; FLT; c-Met/HGFR; TAM Receptor; c-Kit; ROR | Angiogenesis; Metabolism; Tyrosine Kinase/Adaptors |
Cabozantinib hydrochloride (XL184) 是一种有效的泛酪氨酸激酶抑制剂,可抑制 VEGFR2、c-Met、Kit、Axl 和 Flt4(IC50:0.035、1.3、4.6、7 和 6 nM)。 | |||
T6010 |
Idarubicin hydrochloride
盐酸伊达比星,Idamycin,4-demethoxydaunorubicin (NSC256439, 4-DMDR) HCl,4-Demethoxydaunorubicin hydrochloride,Idarubicin HCl,伊达比星盐酸盐,Zavedos |
Topoisomerase; Antibacterial; Autophagy; Antifungal | Autophagy; DNA Damage/DNA Repair; Microbiology/Virology |
Idarubicin hydrochloride (Zavedos) 是一种蒽环类抗白血病药物,能抑制细菌和酵母菌生长,还抑制拓扑异构酶 II,干扰 DNA 复制和 RNA 转录。 | |||
T4261 |
BPR1J-097 hydrochloride (1327167-19-0(free base))
|
FLT | Angiogenesis; Tyrosine Kinase/Adaptors |
BPR1J-097 hydrochloride (1327167-19-0(free base)) 是一种新型小分子 FLT-3抑制剂(IC50=11±7 nM),具有很好的体内抗肿瘤活性。 | |||
T8402 |
Regorafenib Hydrochloride
瑞戈非尼盐酸盐,BAY73-4506 hydrochloride |
Raf; VEGFR; c-RET; PDGFR; Autophagy | Angiogenesis; Apoptosis; Autophagy; MAPK; Tyrosine Kinase/Adaptors |
Regorafenib Hydrochloride (BAY73-4506 hydrochloride) 是一种新型口服多激酶抑制剂,可抑制血管生成、基质和致癌受体酪氨酸激酶,具有强大的临床前抗肿瘤活性。它靶向作用于 VEGFR1/2/3、PDGFRβ、Kit、RET 和 Raf-1,IC50值分别为 13/4.2/46、22、7、1.5 和 2.5 nM。 | |||
T34838 |
Theophylline, 7-(2-oxo-4-piperidinobutyl)-6-thio-, hydrochloride
|
||
Theophylline, 7-(2-oxo-4-piperidinobutyl)-6-thio-, hydrochloride is a bioactive chemical. | |||
T34836 |
Theophylline, 7-(2-(diethylamino)ethyl)-6-thio-, hydrochloride
|
||
Theophylline, 7-(2-(diethylamino)ethyl)-6-thio-, hydrochloride is a bioactive chemical. | |||
T63095 | GNE 220 hydrochloride | ||
GNE 220 (hydrochloride) 是一种有效的、选择性的 MAP4K4 抑制剂 (IC50: 7 nM)。 | |||
T12025 |
MFZ 10-7 hydrochloride
|
GluR | Neuroscience |
MFZ 10-7 hydrochloride is a highly potent and selective negative allosteric modulator of mGluR5 NAM | |||
T61724 | SB 258741 hydrochloride | ||
SB 258741 hydrochloride is a potent antagonist of the 5-HT 7 receptor, designed specifically for studying schizophrenia [1]. | |||
T22091 |
Imiquimod hydrochloride
|
||
Imiquimod hydrochloride (R 837 hydrochloride)是一种免疫反应调节剂,是一种选择性的 toll 样受体 7 (TLR7) 激动剂。Imiquimod hydrochloride 在体内表现出抗病毒和抗肿瘤作用。Imiquimod hydrochloride 可用于外生殖器、肛周疣、癌症和 COVID-19 的研究。 | |||
T11548L |
HCV-IN-7 hydrochloride
|
Others | Others |
HCV-IN-7 hydrochloride is an orally active and potent pan-genotypic HCV NS5A inhibitor (IC50s: 3-47 pM). It shows a superior pan-genotypic profile and a good pharmacokinetic profile coupled with a favorable liver uptake. | |||
T67583 |
Ethyl L-methionate hydrochloride
|
||
Ethyl L-methionate hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T67583,CAS号为 2899-36-7。 | |||
T66353 |
N,N-Dimethylglycine hydrochloride
|
||
N,N-Dimethylglycine hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66353,CAS号为 2491-06-7。 | |||
T63622 | RF9 hydrochloride | ||
RF9 hydrochloride 是有效的、选择性的神经肽 FF 受体 (Neuropeptide FF receptor) 拮抗剂,能够作用于 hNPFF1R (Ki: 58 nM) 和 hNPFF2R (Ki: 7 nM)。 | |||
T19243 |
CMP-5 hydrochloride
|
Others | Others |
CMP-5 hydrochloride is a potent and selective PRMT5 inhibitor, while displays no activity against PRMT1/4/7 enzymes. It selectively blocks S2Me-H4R3 by inhibiting PRMT5 methyltransferase activity on histone preparations. | |||
T65471 | tans-4-Hydroxy-D-proline hydrochloride | ||
tans-4-Hydroxy-D-proline hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65471,CAS号为 142347-81-7。 | |||
T66418 |
L-Threonine methyl ester hydrochloride
|
||
L-Threonine methyl ester hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66418,CAS号为 39994-75-7。 | |||
T66879 |
2-Amino-3-mercaptopropanoic acid hydrochloride xhydrate
|
||
2-Amino-3-mercaptopropanoic acid hydrochloride xhydrate 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66879,CAS号为 96998-61-7。 | |||
T65376 |
2-(tert-Butylamino)acetic acid hydrochloride
|
||
2-(tert-Butylamino)acetic acid hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65376,CAS号为 6939-23-7。 | |||
T65814 | 4-Hydrazinylbenzenesulfonamide hydrochloride | ||
4-Hydrazinylbenzenesulfonamide hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65814,CAS号为 17852-52-7。 | |||
T67608 |
N-(3-Fluorophenyl)piperidin-4-amine hydrochloride
|
||
N-(3-Fluorophenyl)piperidin-4-amine hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T67608,CAS号为 923565-91-7。 | |||
T66533 |
2-Amino-N-(2,2,2-trifluoroethyl)acetamide hydrochloride
|
||
2-Amino-N-(2,2,2-trifluoroethyl)acetamide hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66533,CAS号为 1171331-39-7。 | |||
T66081 |
(S)-1-tert-Butyl 5-methyl 2-aminopentanedioate hydrochloride
|
||
(S)-1-tert-Butyl 5-methyl 2-aminopentanedioate hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66081,CAS号为 34582-33-7。 | |||
T65425 |
2-(Methylamino)acetic acid hydrochloride
|
||
2-(Methylamino)acetic acid hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65425,CAS号为 637-96-7。 | |||
T67214 |
2-((Dimethylamino)methyl)cyclohexanone hydrochloride
|
||
2-((Dimethylamino)methyl)cyclohexanone hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T67214,CAS号为 42036-65-7。 | |||
T66230 |
trans-4-Dimethylaminocrotonic acid hydrochloride
|
||
trans-4-Dimethylaminocrotonic acid hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66230,CAS号为 848133-35-7。 | |||
T78150 |
USP7-IN-10 hydrochloride
|
||
USP7-IN-10 hydrochloride (compound 1)是一种高效USP7抑制剂,具有13.39 nM的IC50值。 | |||
T66037 |
(R)-Tetrahydropapaverine hydrochloride
|
||
(R)-Tetrahydropapaverine hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66037,CAS号为 54417-53-7。 | |||
T71764 | YM 298198 Hydrochloride | ||
YM 298198 Hydrochloride is a non-competitive antagonist with high affinity and selectivity for mGlu1 receptors (Ki = 19 nM). YM 298198 Hydrochloride is inactive at other mGlu receptor subtypes (mGlu2-7), ionotropic receptors and glutamate transporters (IC50 > 10 μM). It inhibits glutamate-induced IP production more potently than CPCCOEt (IC50 values are 16 nM and 6.3 μM respectively). | |||
T66383 | 3-(Piperidin-4-yl)benzo[d]oxazol-2(3H)-one hydrochloride | ||
3-(Piperidin-4-yl)benzo[d]oxazol-2(3H)-one hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66383,CAS号为 162045-54-7。 | |||
T13157L | TG 100801 Hydrochloride | VEGFR | Angiogenesis; Tyrosine Kinase/Adaptors |
TG 100801 Hydrochloride is a prodrug to treat age-related macular degeneration. TG 100572 is a inhibitor of multi-targeted kinase(IC50s of 2, 7, 2, 16, 13, 5, 0.5, 6, 0.1, 0.4, 1, 0.2 for VEGFR1, VEGFR2, FGFR1, FGFR2, PDGFRβ, Fgr, Fyn, Hck, Lck, Lyn, Src, | |||
T64682 | 2-Amino-6-(propylamino)-5,6-dihydrobenzo[d]thiazol-7(4H)-one hydrochloride | ||
2-Amino-6-(propylamino)-5,6-dihydrobenzo[d]thiazol-7(4H)-one hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T64682。 | |||
T36231 |
rac-7-hydroxy Propranolol (hydrochloride)
|
||
rac-7-hydroxy Propranolol (hydrochloride) is a ring-hydroxylated isomer and metabolite of propranolol that is an antagonist at β-adrenergic receptors (0.95 potency relative to propranolol). It also demonstrates potent vasodilator activity (0.20 potency relative to propranolol; pA2 = 7.58). | |||
T66095 |
5-Methyl-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridine-2-carboxylic acid hydrochloride
|
||
5-Methyl-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridine-2-carboxylic acid hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66095,CAS号为 720720-96-7。 | |||
T64405 |
6-Methyl-1,3-dihydrofuro[3,4-c]pyridin-7-ol hydrochloride
|
||
6-Methyl-1,3-dihydrofuro[3,4-c]pyridin-7-ol hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T64405,CAS号为 1006-21-9。 | |||
T65519 |
(6R,7R)-4-Methoxybenzyl 7-amino-3-(chloromethyl)-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylate hydrochloride
|
||
(6R,7R)-4-Methoxybenzyl 7-amino-3-(chloromethyl)-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylate hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65519,CAS号为 113479-65-5。 | |||
T13156L |
TG 100572 Hydrochloride
|
VEGFR; FGFR; PDGFR; Src | Angiogenesis; Tyrosine Kinase/Adaptors |
TG 100572 Hydrochloride 是一种多靶点激酶抑制剂,能够抑制受体酪氨酸激酶和Src 激酶。 | |||
T77873 |
NH2-bicyclo[1.1.1]pentane-7-MAD-MDCPT hydrochloride
|
Topoisomerase | DNA Damage/DNA Repair |
NH2-bicyclo[1.1.1]pentane-7-MAD-MDCPT(化合物I)盐酸盐是一种通过偶联抗体实现靶向细胞传递的拓扑异构酶I抑制剂,显示出优良的体内外ADC活性。 | |||
T77865 |
Tetrazine-PEG7-amine hydrochloride
|
||
Tetrazine-PEG7-amine hydrochloride 为含有7个单元聚乙二醇(PEG)的可降解ADC链接剂,适用于抗体偶联药物(ADCs)的合成。 | |||
T68262 | AEG40826 | ||
AEG40826 (HGS1029) is the hydrochloride salt of a small-molecule inhibitor of IAP (Inhibitor of Apoptosis Protein) family proteins with potential antineoplastic activity. IAP inhibitor HGS1029 selectively inhibits the biological activity of IAP proteins, which may restore apoptotic signaling pathways; this agent may work synergistically with cytotoxic drugs to overcome tumor cell resistance to apoptosis. IAPs are overexpressed by many cancer cell types, suppressing apoptosis by binding and inhib... | |||
T35875 | CCG258208 hydrochloride | ||
GRKs-IN-1 hydrochloride, Compound 14as, has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50=130 nM) and GRK5 (IC50=7.1 μM).GRKs-IN-1 hydrochloride is a derivative 14as of paroxetine, shows a 100-fold improvement in cardiomyocyte contractility assays over paroxetine[1]. [1]. Waldschmidt HV, et al. Structure-Based Design of Highly Selective and Potent G Protein-Coupled Receptor Kinase 2Inhibitors Based on Paroxetine. J Med Chem. 2017 Apr 13;60(7):305... | |||
T70235 |
Cemadotin hydrochloride
|
||
Cemadotin hydrochloride is the salt from of Cemadotin (free base), also known as, LU103793, a mitosis inhibitor potentially for the treatment of solid tumours. Cemadotin is also a synthetic derivative of Dolastatin 15, an antiproliferative compound which was isolated from the mollusk Dolabella auricularia. Like Dolastatin 15, LU103793 is highly cytotoxic in vitro (IC50 = 0.1 nM). LU103793 inhibits microtubule polymerization in a concentration-dependent manner (IC50 = 7 microM). Treatment with ... |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1400 |
Demeclocycline hydrochloride
地美环素,Declomycin,Clortetrin,盐酸地美环素,Detravis,Demeclocycline HCl |
ribosome; Antibacterial; Antibiotic | Microbiology/Virology |
Demeclocycline hydrochloride (Declomycin) 是四环素类抗生素,可治疗粉刺,莱姆病和支气管炎。 | |||
T0486L |
Irinotecan Hydrochloride
盐酸伊立替康,伊立替康盐酸盐,Camptothecin 11 hydrochloride,CPT-11 hydrochloride |
Topoisomerase; Autophagy | Autophagy; DNA Damage/DNA Repair |
Irinotecan Hydrochloride (CPT-11 hydrochloride) 是喜树碱半合成衍生物的盐酸盐,是一种拓扑异构酶 I 抑制剂,可研究结肠癌和直肠癌。 |